99% Tianeptine sodium cusbo CAS 30123-17-2
Tilmaamid
ITEM | HEERKA | NATIIJO |
Muuqashada | Caddaan ilaa budo huruud ah | Budada crystalline cad |
Solubility | Si xor ah ugu milmay biyaha iyo methanol iyo dichloromethane | waafaqsan |
Aqoonsiga | By IR, Si loo waafajiyo heerka shaqada | waafaqsan |
(2) Waxay bixisaa falcelin soodhiyam ah | waafaqsan | |
wasakhda A | ≤0.1% | Lama ogaan |
Iskudhisyada la xidhiidha | Mid kasta oo ugu badan oo wasakh ah≤0.1% | 0.060% |
Wadarta wasakhda≤0.4% | 0.36% | |
Xalalka Hadhaaga ah (GC) | Acetidin≤ 0.5% | ND |
Dichloromethane≤ 0.06% | ND | |
Methanol≤ 0.3% | ND | |
Acetone ≤ 0.5% | 0.29% | |
Acetonitrile≤0.041% | 0.022% | |
Ethanol≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Biyo | ≤ 5.0% | 3.8% |
Qiimaynta (HPLC) | 99.0% -101.0% (oo ku salaysan anhydrousbasis) | 99.70% |
Codsiga
Tianeptine sodiumcusbowaa tricyclic antidepressant.Nidaamkeeda ka hortagga niyad-jabka way ka duwan tahay kuwa dhaqameed ee tricyclic antidepressants.Waxay kordhin kartaa dib-u-qaadista 5-HT ee dillaaca synaptik.Saamaynta HT neuronal conduction.Wax xidhiidh ah uma laha choline ama adrenergic reseptors.Waxtarka ka hortagga niyad-jabka wuxuu la mid yahay kan tricyclics, laakiin dulqaadku wuu ka fiican yahay kan tricyclics.Daawaynta niyad-jabka khafiifka ah, dhexdhexaadka ah ama daran, neurogenic iyo niyad-jabka falcelinta, walaaca iyo niyad-jabka jirka, gaar ahaan raaxo-darrada caloosha iyo mindhicirka, iyo walaaca iyo niyad-jabka bukaanka ku-tiirsan khamriga inta lagu jiro bixitaanka.